Synthesis of new multitarget-directed ligands containing thienopyrimidine nucleus for inhibition of 15-lipoxygenase, cyclooxygenases, and pro-inflammatory cytokines

Faculty Pharmacy Year: 2023
Type of Publication: ZU Hosted Pages:
Authors:
Hend Kather Abdelhakem Elhamalawy
Journal: ُEuropean Journal of Medicinal Chemistry ُElsevier Volume:
Keywords : Synthesis , , multitarget-directed ligands containing thienopyrimidine nucleus    
Abstract:
A new series of thieno[2,3-d]pyrimidine derivatives 4, 5, 6a-o, and 11 was designed and synthesized starting from cyclohexanone under Gewald condition with the aim to develop multitarget-directed ligands (MTDLs) having anti-inflammatory pro
    
     
 
       

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Department Related Publications

  • Alsayed Mohamed Mansour Lashen , "Synthesisis Of Certain Condensed Pyrimidines", لايوجد, 1900 More
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  • Rania Hamdy Ahmed Badawi, " Synthesis Of Novel 2-Sbstituted Quinaline -4-Carboxylic Acid Derivatives For Potential Biological Activity", لايوجد, 1900 More
  • Samy Megahed Ibrahiem Elsayed Sakr, "Synthesis Of Certain -4-Quinazolones Likely To Possess Pharmacological Activity", لايوجد, 1900 More
  • Samy Megahed Ibrahiem Elsayed Sakr, "ٍSynthesis And Biological Activity Of Some Novel Heterocyclic Compounds Containing Sulphar Of Pharmaceutical Interest ", لايوجد, 1900 More
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