Novel benzenesulfonamide and 1,2-benzisothiazol-3(2H)-one-1,1-dioxide derivatives as potential selective COX-2 inhibitors

Faculty Pharmacy Year: 2019
Type of Publication: ZU Hosted Pages: 372-382
Authors:
Tarek Mohamed Salah Rashad
Journal: European Journal of Medicinal Chemistry ELSEVIER FRANCE-EDITIONS SCIENTIFIQUES MEDICALES ELSEVIER Volume:
Keywords : Novel benzenesulfonamide , 1,2-benzisothiazol-3(2H)-one-1,1-dioxide derivatives , potential selective    
Abstract:
Two new series of 1,2-benzisothiazol-3(2H)-one-1,1-dioxide derivatives containing either five membered heterocyclic rings or aryl hydrazones were synthesized and evaluated for their in vitro COX-1/COX-2 inhibitory activity. In vivo anti-inf
    
     
 
       

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Department Related Publications

  • Zakareyah Kamel Abdelsamie, "Synthesis of some novel s-triazolo[3,4-b]-1,3,4-thiadiazole derivatives as antiinflammatory agents", Proceedings of XXI conference of Pharmaceutical Sciences, 1990 More
  • Zakareyah Kamel Abdelsamie, "Synthesis and antibacterial activity of novel benzothiazole, benzimidazole, imidazolidine and imidazo-[2,1-b]-1,3,4-thiadiazole derivatives", Bull. Fac. Pharm. Cairo Univ, 1994 More
  • Etedaal Hassan Mohamed Abdulaal, "15. Application of Reductive Nitrosation in Synthesis of Pyrroloquinoxalines as Antimicrobial Agents", لايوجد, 1900 More
  • Hanan Abdelraziek Abdelfattah Ali Hamied, "Synthesis of certain quinazolinone derivatives of pharmaceutical interest", 2024 More
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