Synthesis, antibacterial properties and 2D-QSAR studies of quinolone-triazole conjugates

Faculty Pharmacy Year: 2018
Type of Publication: ZU Hosted Pages: 1524-1534
Authors:
Amany Mohamed Mohamed Elmahmoudy Sanger
Journal: European Journal of Medicinal Chemistry ElSevier Volume: 2018
Keywords : Synthesis, antibacterial properties , 2D-QSAR studies , quinolone-triazole    
Abstract:
A set of 1,2,3-triazole incorporated quinolone antibiotic conjugates 10–15, 17–19 were synthesized via microwave assisted click chemistry technique. Some of the aryl-substituted conjugates 17–19 show promising antibacterial properties again
    
     
 
       

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