Synthesis, biological evaluation, and radioiodination of halogenated closo-carboranylthymidine analogues

Faculty Science Year: 2011
Type of Publication: ZU Hosted Pages:
Authors:
Ahmed Khalil Elsayed Khalil
Journal: Nucleosides, Nucleotides and Nucleic Acids ACS Volume:
Keywords : Synthesis, biological evaluation, , radioiodination , halogenated closo-carboranylthymidine    
Abstract:
The synthesis and initial biological evaluation of 3-carboranylthymidine analogues (3CTAs) that are (radio)halogenated at the closo-carborane cluster are described. Radiohalogenated 3CTAs have the potential to be used in the radiotherapy an
    
     
 
       

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