A Series of Pyridines and Pyridine Based Sulfa-Drugs as Antimicrobial Agents: Design, Synthesis and Antimicrobial Activity1

Faculty Science Year: 2017
Type of Publication: ZU Hosted Pages: 2401-2408
Authors:
Ahmed Heussein Mostafa
Journal: Russian Journal of General Chemistry ٍspringer Volume: 87
Keywords : , Series , Pyridines , Pyridine Based Sulfa-Drugs as Antimicrobial    
Abstract:
Herein, we report a series of pyridines and their sulfa drug derivatives as antimicrobial agents. Regioselective alkylation followed by hydrozinolysis of 2-pyridone 1 gave the target compounds 2 and 3. Compound 3 was cyclized with acetyla
    
     
 
       

Author Related Publications

  • Ahmed Heussein Mostafa, "Evaluation of the Curative and Protective Role of Fresh Chicory Juice in Treatment of Hepatic Fibrosis in Male Albino Rats", Scoups, 2021 More
  • Ahmed Heussein Mostafa, "Efficient biocontrol of Spodoptera littoralis by Aspergillus nidulans, an endophyte of Lantana camara", ٍSpringer, 2020 More
  • Ahmed Heussein Mostafa, "Synthesis and Biological Evaluation of Glycosides and AcyclicNucleosides Derived 2-Oxonicotinonitriles", Wiely, 2019 More
  • Ahmed Heussein Mostafa, "Novel Triazole-, Oxadiazole-, and Pyrazole-Nicotinonitrile Hybrids: Synthesis, DFT Study, Molecular Docking, and Antimicrobial Activity", ٍSpringer, 2022 More
  • Ahmed Heussein Mostafa, "Synthesis and biological evaluation of 2-Oxo/thioxoquinoxaline and 2-Oxo/thioxoquinoxaline-based nucleoside analogues", EBSCO, 2016 More

Department Related Publications

  • Mohamed Gamal Helmy Mohamed Abdelwahed, "Electronic Properties of Organic Complexes. 2. Reactive Azodyes", Spain, 1993 More
  • Mohamed Gamal Helmy Mohamed Abdelwahed, "Electrical Behaviour of some Azodye Mixed Ligand with Gd3+ and Er3+. b", Peru, 1994 More
  • Atef Mohamed AbdelHamid Ali Hassn, "heterocyclization of thiouracil derivative: synthesis of thiazolopyrimidines, tetrazolopyrimidines and triazolopyrimidines of potential biological activity", elsevier, 2015 More
  • Mohammed Aref Awad Allah Abu Zyd, "Synergistic positive effects of nano barium silicate on the hydration rate and phase composition of alkali-activated slag", Elsevier, 2022 More
  • Ahmed Abdelmoniem Ahmed Amer, "Synthesis and characterization of some calcium aluminate phases from nano-size starting materials", 0366-3175/© 2020 SECV. Published by Elsevier Espana, ˜ S.L.U, 2020 More
Tweet